articleOrganic Process Research & DevelopmentNov 15, 2015Closed access

Large-Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals

Gilead Sciences (United States) · Pfizer (United States)

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Abstract

This review showcases various coupling reagents which have been implemented specifically for large-scale amide synthesis via the condensation of an acid and amine, while highlighting the benefits and drawbacks of each reagent on an industrial scale.

Citation impact

793
total citations
FWCI
18.97
Percentile
100%
References
464
Citations per year

Authors

3

Topics & keywords

Keywords
  • Reagent
  • Amide
  • Amine gas treating
  • Combinatorial chemistry
  • Scale (ratio)
  • Coupling (piping)
  • Chemistry
  • Condensation
UN Sustainable Development Goals
  • Industry, innovation and infrastructure
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