articleProceedings of the National Academy of SciencesMar 28, 2016BRONZE OA

Stimuli-responsive clustered nanoparticles for improved tumor penetration and therapeutic efficacy

University of Science and Technology of China · Georgia Institute of Technology · +3 more institutions

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Abstract

A principal goal of cancer nanomedicine is to deliver therapeutics effectively to cancer cells within solid tumors. However, there are a series of biological barriers that impede nanomedicine from reaching target cells. Here, we report a stimuli-responsive clustered nanoparticle to systematically overcome these multiple barriers by sequentially responding to the endogenous attributes of the tumor microenvironment. The smart polymeric clustered nanoparticle (iCluster) has an initial size of ∼100 nm, which is favorable for long blood circulation and high propensity of extravasation through tumor vascular fenestrations. Once iCluster accumulates at tumor sites, the intrinsic tumor extracellular acidity would…

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