reviewSignal Transduction and Targeted TherapyJun 24, 2022GOLD OA

Targeting signaling pathways in prostate cancer: mechanisms and clinical trials

East China Normal University · Shanghai Changzheng Hospital · +5 more institutions

PubMed
Indexed incrossrefdoajpubmed

Abstract

Abstract Prostate cancer (PCa) affects millions of men globally. Due to advances in understanding genomic landscapes and biological functions, the treatment of PCa continues to improve. Recently, various new classes of agents, which include next-generation androgen receptor (AR) signaling inhibitors (abiraterone, enzalutamide, apalutamide, and darolutamide), bone-targeting agents (radium-223 chloride, zoledronic acid), and poly(ADP-ribose) polymerase (PARP) inhibitors (olaparib, rucaparib, and talazoparib) have been developed to treat PCa. Agents targeting other signaling pathways, including cyclin-dependent kinase (CDK)4/6, Ak strain transforming (AKT), wingless-type protein (WNT), and epigenetic marks, have…

Citation impact

250
total citations
FWCI
34.30
Percentile
100%
References
594
Citations per year

Authors

6

Topics & keywords

Keywords
  • Olaparib
  • Prostate cancer
  • Enzalutamide
  • Medicine
  • Cancer research
  • Pembrolizumab
  • Androgen receptor
  • Clinical trial
UN Sustainable Development Goals
  • Good health and well-being
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Funding