articleACS NanoFeb 3, 2025Closed access

Cuproptosis-Inducing Functional Nanocomposites for Enhanced and Synergistic Cancer Radiotherapy

Shanghai Jiao Tong University · Shanghai Chest Hospital · +7 more institutions

PubMed
Indexed incrossrefpubmed

Abstract

Radiotherapy is crucial in local cancer management and needs advancements. Tumor cells elevate intracellular copper levels to promote growth and resist radiation; thus, targeted copper delivery to mitochondria could enhance radiotherapy by inducing cuproptosis in tumor cells. In this study, we engineered a multifunctional nanoliposome complex, termed Lipo-Ele@CuO2, which encapsulates both copper peroxide (CuO2) and the copper chelator elesclomol, which can delivery Cu ions to the mitochondria. The Lipo-Ele@CuO2 complex induces mitochondria-mediated cuproptosis in tumor cells and synergistically enhances the efficacy of radiotherapy. CuO2 acts as a copper donor and exhibits inherent sensitivity to acidic…

Citation impact

42
total citations
FWCI
21.96
Percentile
100%
References
57
Citations per year

Authors

10

Topics & keywords

Keywords
  • Radiation therapy
  • Cancer research
  • Cancer cell
  • Tumor microenvironment
  • Mitochondrion
  • Intracellular
  • Radioresistance
  • Chemistry
No related works found for this paper.

Funding